BDBM10887 Sulfamate 7::Topiramate (TPM)::US11535599, Example topiramate::[(1R,2S,6S,9R)-4,4,11,11-tetramethyl-3,5,7,10,12-pentaoxatricyclo[7.3.0.0^{2,6}]dodecan-6-yl]methyl sulfamate
SMILES CC1(C)O[C@@H]2CO[C@@]3(COS(N)(=O)=O)OC(C)(C)O[C@H]3[C@@H]2O1
InChI Key InChIKey=KJADKKWYZYXHBB-XBWDGYHZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 10887
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of human recombinant CA5A after 15 mins by CO2 hydration stopped flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of human carbonic anhydrase 5AMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of human recombinant CA5A by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of human recombinant CA5A by CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of full length human carbonic anhydrase 5a preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of human recombinant CA5A mitochondrial isoform by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nM ΔG°: -9.82kcal/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of human carbonic anhydrase 5A after 15 mins by stopped flow carbon dioxide hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKi: 6.30E+4nMAssay Description:Inhibition of full length human recombinant mitochondrial carbonic anhydrase 5A pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Ecole Nationale Sup£Rieure De Chimie De Montpellier
Curated by ChEMBL
Affinity DataKd: 25.4nMAssay Description:Inhibition of human carbonic anhydrase 5AMore data for this Ligand-Target Pair